TripSit · Fasoracetam

正文中文为机器翻译，仅供参考；专业内容以折叠的原文为准。

详情

分类

research-chemical 促智剂 tentative

后遗时间

1-6 小时

剂量

口服

常规

5-10mg

轻度

2.5-5mg

强效

10-25mg.

持续时间

4-8 小时

起效时间

10-45 分钟

名称

fasoracetam

通用名

Fasoracetam

属性

后遗效应

1–6 小时.

分类

research-chemical 促智剂 tentative

剂量

Low: 2.5-5mg Common: 5-10mg Strong: 10-25mg.

持续

4–8 小时.

起效

10–45 分钟.

摘要

A substance in the racetam family. The drug has been shown to reverse memory impairment caused by baclofen, a potent GABA(B) agonist. It additionally has been shown to inhibit baclofen-induced suppression of cyclic AMP formation. The drug is indicated to have a type of GABA(B) antagonistic action. The drug has been shown to reverse high-affinity choline uptake induced by electrolytic lesions of the basal forebrain and pentobarbital anesthesia. It additionally has indications of having antidepressant activity and through repeated dosage, up-regulation of GABA(B) receptors. Notably, the indications of antidepressant activity were noted to be isolated, not affecting monoamine uptake nor central monoaminergic transmission. In addition to not affecting B-adrenoceptors and 5HT2 receptors. Clinical studies of the drug have failed to show statistical signifigance in treatments for a variety of disorders, but further clinical trials are underway.